Targets to Therapeutics in Pancreatic Cancer


NIH funded program project grant

VON HOFF, DANIEL D.

Grant Number: P01CA109552


Our Team Pubs Pancreatic Neoplasm Clinical Trials Pubmed Review Articles  Case Reports


Antwi K, Hostetter G, Demeure MJ, Decker GA, Ruiz Y, Sielaff T, Koep L, Lake DF.  Analysis of human plasma peptidome reveals potential biomarkers for pancreatic cancer. J Prot Res (in press).

 

*Azorsa DO, Gonzales IM, Basu GD, Choudhary A, Arora S, Bisanz KM, Kiefer JA, Henderson MC, Trent JM, Von Hoff DD, Mousses S. Synthetic lethal RNAi screening identifies sensitizing targets for gemcitabine therapy in pancreatic cancer. J Transl Med. 2009 Jun 11;7:43. PMCID: PMC2702280.

 

*Baker AF, Dragovich T, Tate WR, Ramanathan RK, Roe D, Hsu DH, Kirkpatrick DL, Powis G. The antitumor thioredoxin-1 inhibitor PX-12 (1-methylpropyl 2-imidazolyl disulfide) decreases thioredoxin-1 and VEGF levels in cancer patient plasma. J Lab Clin Med 2006;147:83-90. PMCID: PMC1432091


*Baker AF, Koh MY, Williams RR, James B, Wang H, Tate WR, Gallegos A, Von Hoff DD, Han H, Powis G. Identification of thioredoxin-interacting protein 1 as ahypoxia-inducible factor 1alpha-induced gene in pancreatic cancer. Pancreas. 2008Mar;36(2):178-86.

 

*Baker AF, Landowski T, Dorr R, Tate WR, Gard JM, Tavenner BE, Dragovich T, Coon A, Powis, G. The antitumor agent imexon activates antioxidant gene expression: evidence for an oxidative stress response. Clin Cancer Res 2007;13:3388-3394.

 

*Balagurunathan Y, Morse DL, Hostetter G, Shack S, Stafford P, Vijayalashimi S, Pearson J, Trissal M, Demeure MJ, Bittner M, Gilles RJ, Han H.  Gene expression profiling based identification of cell surface targets for developing multimeric ligands in pancreatic cancer. Mol Cancer Ther 2008;7(9):3071-3080. PMCID: 2567866 [Available on 2009/09/01].

 

Chen S, Auletta T, Dovirak O, Hutter C, Kuntz K, El-Ftesi S, Kendall J, Han H, Von Hoff DD, Ashfaq R, Maitra A, Iacobuzio-Donahue CA, Hruban RH, Lucito R. Copy number alterations in pancreatic cancer identify recurrent PAK4 amplification. Cancer Biol Ther. 2008;7(11).

 

*Colvin J, Monine MI, Faeder JR, Hlavacek WS, Von Hoff DD, Posner, RG. Simulation of large-scale rule-based models. Bioinformatics. 2009 Apr ;25(7):910-7. PMCID: PMC2660871 [Available on 2010/04/01]

 

*Dragovich T, Burris H 3rd, Loehrer P, Von Hoff DD, Chow S, Stratton S, Green S, Obregon Y, Alvarez I, Gordon M.  Gemcitabine plus celecoxib in patients with advanced or metastatic pancreatic adenocarcinoma: results of a phase II trial. Am J Clin Oncol. 2008 Apr;31(2):157-62.

 

Dragovich T, Huberman M, Von Hoff DD, Rowinsky EK, Nadler P, Wood D, Hamilton M, Hage G, Wolf J, Patnaik A.Erlotinib plus gemcitabine in patients with unresectable pancreatic cancer and other solid tumors: phase IB trial. Cancer Chemother Pharmacol. 2007 Jul;60(2):295-303. Epub 2006 Dec 6.

 

*Henderson MC, Shaw YJ, Wang H, Han H, Hurley LH, Flynn G, Dorr RT, Von Hoff DD. UA62784, a novel inhibitor of centromere protein E kinesin-like protein. Mol Cancer Ther. 2009 Jan;8(1):36-44. PMCID: PMC2634858.

 

Hu B, Matthew Fricke G, Faeder JR, Posner RG, Hlavacek WS. GetBonNie for building, analyzing and sharing rule-based models. Bioinformatics. 2009 Jun 1;25(11):1457-60. PMCID: PMC2682519 [Available on 2010/06/01]

 

Jordan BF, Black K, Robey IF, Runquist M, Powis G, Gillies R. Metabolite changes in HT-29 xenografts tumors following HIF-1” inhbition with PX-478 as studied by MR spectroscopy in vivo and ex vivo. NMR Biomed 2005;18:1-10.

 

Kahlem P, Newfeld SJ. Informatics approaches to understanding TGFβ pathway regulation.  Development 2009;136 (in press). 

 

Kiefer J, Yin HH, Que QQ, Mousses S. High-Throughput siRNA Screening as a Method of Perturbation of Biological Systems and Identification of Targeted Pathways Coupled with Compound Screening. Methods Mol Biol. 2009;563:275-87.

 

Koh MY, Darnay BG, Powis G. HAF, a novel E3-ubiquitin ligase binds to and ubiquitinates HIF-1α leading to its pVHL- and oxygen-independent degradation. Mol Cell Biol, 2008;28(23):7081-7095. PMCID: PMC2593390


Koh M, Powis G. HAF, the new player in oxygen-independent HIF-1α degradation. Cell Cycle. 2009 May 1;8(9):1359-66. PMCID: PMC2700049

 

Koh, M Y, Spivak-Kroizman, T.R and Powis, G. Inhibiting the Hypoxia Response for Cancer Therapy: The New Kid on the Block.  Clin Cancer Res 2009;15(19) (in press). 

 

Koh MY, Spivak-Kroizman T, Venturini S, Welsh S, Williams R, Powis G. Molecular mechanisms for the activity of PX-478, an antitumor inhibitor of the hypoxia inducible factor-1a (HIF-1a). Mol Cancer Ther 2008;7:90-100.

 

Koh MY, Taly R, Spivak-Kroizman TR, Powis G. HIF-1 regulation: not so easy come easy go. Trends Biochem Sci. 2008 Nov;33(11):526-34.


Kuuselo R, Savinainen K, Azorsa DO, Basu GD, Karhu R, Tuzmen S, Mousses S, Kallioniemi A. Intersex like (IXL) is a cell survival regulator in pancreatic cancer with 19q13 amplification. Cancer Res 2007;67(5):1943-1949.

 

Laurila E, Savinainen K, Kuuselo R, Karhu R, Kallioniemi A. Characterization of the 7q21-q22 Amplicon Identifies ARPC1A, a Subunit of the Arp2/3 Complex, as a Regulator of Cell Migration and Invasion in Pancreatic Cancer. Genes Chromosomes Cancer. 2009 Apr;48(4):330-9.

 

*Mahadevan D, Dreisbach L, Kristadja T, Williams D, Obregon Y, Kurtin S, Von Hoff D. Phase I study of fixed dose gemcitabine combined with epirubicin in patients with advanced solid malignancies. Am J Clin Oncol. 2009 Jul 10. [Epub ahead of print]

 

*Mahadevan D, Powis G, Mash EA, George B, Gokhale VM, Zhang S, Shakalya K, Du-Cuny L, Berggren M, Ali MA, Jana U, Ihle N, Moses S, Franklin C, Narayan S, Shirahatti N, Meuillet EJ. Discovery of a novel class of AKT pleckstrin homology domain inhibitors. Mol Cancer Ther 2008;7(9):2621-32. PMCID: PMC2727864

 

*Mahadevan D, Von Hoff DD. Tumor-stroma interactions in pancreatic ductal adenocarcinoma. Mol Cancer Ther. 2007 Apr;6(4):1186-97.

 

Monine MI, Posner RG, Savage PB, Faeder JR, Hlavacek WS Modeling multivalent ligand interactions with steric constraints on configurations of cell-surface aggregates. Biophysical Journal  2009 (in press).

 

*Mount DW, Pandey R. Using bioinformatics and genome analysis for new therapeutic interventions. Mol Cancer Ther. 2005;4:1636-43.

 

Mount DW. Cold Spring Harbor Protocols: Bioinformatics and Genomics.  Cold Spring Harbor Press, 2009 Cold Spring Harbor, NY.

 

*Mousses S., Kiefer J., Von Hoff D., Trent J.  Using BioIntelligence to Search the Cancer Genome: An Epistemological Perspective on Knowledge Recovery Strategies to Enable Precision Medical Genomics.  Oncogene. 2009 (in press).

 

Powis G, Kirkpatrick DL.  Thioredoxin signaling as a target for cancer therapy. Curr Opin Pharmacol. 2007;7(4):392-397.

*Ramanathan RK, Kirkpatrick DL, Belani CP, Friedland D, Green SB, Chow HH, Cordova CA, Stratton SP, Sharlow ER, Baker A, Dragovich TA.  Phase I pharmacokinetic and pharmacodynamic study of PX-12, a novel inhibitor of thioredoxin-1, in patients with advanced solid tumors. Clin Cancer Res 2007;13:2109-2114.

 

Riley CJ, Engelhardt KP, Saldanha JW, Qi W, Cooke LS, Zhu Y, Narayan ST, Shakalya K, Croce KD, Georgiev IG, Nagle RB, Garewal H, Von Hoff DD, Mahadevan D. Design and activity of a murine and humanized anti-CEACAM6 single-chain variable fragment in the treatment of pancreatic cancer.  Cancer Res. 2009 Mar 1;69(5):1933-40. Epub 2009 Feb 24.

 

Schwartz DL, Thitai-Kumar A, He Y, Williams R, Lemos R, Oh J, Bankson J, Jackson E, Volgin A, Soghomonyan S, Mukhopadhay U, Alauddin M, Kuno N, Krishnan S, Bornman W, Gelovani J, Powis G. The selective HIF-1 inhibitor PX-478 enhances in vivo tumor radio-curability through tumor stromal effects. Mol Cancer Ther. 2009 Apr;8(4):947-58.

 

*Shaw A, Henderson MC, Flynn G, Samulitis B, Han H, Stratton S, Chow HH, Hurley LH, Dorr RT. Characterization of Novel Diaryloxazole-Based Compounds as Potential Agents to Treat Pancreas Cancer. J Pharmacol Exp Ther. 2009 Aug 5. [Epub ahead of print]

 

Stephens BJ, Han H, Gokhale V, Von Hoff DD. PRL phosphatases as potential molecular targets in cancer. Mol Cancer Ther. 2005 Nov;4(11):1653-61. Review.


*Stephens B, Han H, Hostetter G, Demeure MJ, Von Hoff DD. Small interfering RNA-mediated knockdown of PRL phosphatases results in altered Akt phosphory-lation and reduced clonogenicity of pancreatic cancer cells. Mol Cancer Therapeutics 2008;7(1):202-210.

 

Tari L, Baral C, Kim S. Fuzzy c-means clustering with prior biological knowledge. J Biomed Inform. 2009 Feb;42(1):74-81. PMCID: PMC2673503

 

*Tuzmen S, Kiefer J, Mousses S. Validation of short interfering RNA knockdowns by quantitative real-time PCR.  Methods Mol Biol. 2007;353:177-203.

 

Von Hoff DD. What's new in pancreatic cancer treatment pipeline? Best Pract Res Clin Gastroenterol. 2006 Apr;20(2):315-26.

 

*Von Hoff DD, Korn R, Mousses S. Pancreatic cancer—could it be that simple? A different context of vulnerability. Cancer Cell. 2009 Jul 7;16(1):7-8.

 

*Wang H, Han H, Mousses S, Von Hoff DD. Targeting loss-of-function mutations in tumor-suppressor genes as a strategy for development of cancer therapeutic agents. Seminars in Oncology 2006;33:513-520.

 

Wang H, Han H, Von Hoff DD. Identification of an agent selectively targeting DPC4 (deleted in pancreatic cancer locus 4)-deficient pancreatic cancer cells. Cancer Res 2006;66(19):9722-30.

 

Wang H, Stephens B, Von Hoff DD, Han H. Identification and Characterization of a Novel Anticancer Agent With Selectivity Against Deleted in Pancreatic Cancer Locus 4 (DPC4)-Deficient Pancreatic and Colon Cancer Cells. Pancreas. 2009 Jul;38(5):551-7.

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